Pharmacokinetics After oral ingestion, Pregabalin is rapidly absorbed (Tmax 1.3 hr) Bioavailability is >90% and independent of dose Pregabalin is NOT protein bound Vd is 0.4 L/kg Serum pregabalin concentrations are linearly related to dosage Pregabalin is NOT metabolized Pregabalin is primarily excreted unchanged in urine (98%) with a clearance…